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-Structure paper
Title | Ligand-Based Design of Allosteric Retinoic Acid Receptor-Related Orphan Receptor gamma t (ROR gamma t) Inverse Agonists. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 241-259, Year 2020 |
Publish date | Jul 17, 2019 (structure data deposition date) |
![]() | Meijer, F.A. / Doveston, R.G. / de Vries, R.M.J.M. / Vos, G.M. / Vos, A.A.A. / Leysen, S. / Scheepstra, M. / Ottmann, C. / Milroy, L.G. / Brunsveld, L. |
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Methods | X-ray diffraction |
Resolution | 1.61 Å |
Structure data | ![]() PDB-6sal: |
Chemicals | ![]() ChemComp-L3E: ![]() ChemComp-HOH: |
Source |
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![]() | GENE REGULATION / Nuclear Receptor / Allosteric / Inverse Agonist / Inhibitor |