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-Structure paper
Title | Fast Iterative Synthetic Approach toward Identification of Novel Highly Selective p38 MAP Kinase Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 10757-10782, Year 2019 |
Publish date | Aug 1, 2019 (structure data deposition date) |
![]() | Rohm, S. / Berger, B.T. / Schroder, M. / Chaikuad, A. / Winkel, R. / Hekking, K.F.W. / Benningshof, J.J.C. / Muller, G. / Tesch, R. / Kudolo, M. ...Rohm, S. / Berger, B.T. / Schroder, M. / Chaikuad, A. / Winkel, R. / Hekking, K.F.W. / Benningshof, J.J.C. / Muller, G. / Tesch, R. / Kudolo, M. / Forster, M. / Laufer, S. / Knapp, S. |
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Methods | X-ray diffraction |
Resolution | 1.6 - 1.95 Å |
Structure data | ![]() PDB-6sfi: ![]() PDB-6sfj: ![]() PDB-6sfk: |
Chemicals | ![]() ChemComp-LB5: ![]() ChemComp-HOH: ![]() ChemComp-LBB: ![]() ChemComp-EDO: ![]() ChemComp-LB8: |
Source |
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![]() | TRANSFERASE / p38a / MAPK / MAPK14 / kinase inhibitor / Structural Genomics / Structural Genomics Consortium / SGC |