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-Structure paper
| Title | An isoform-selective inhibitor of tropomyosin receptor kinase A behaves as molecular glue. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 30, Page 126775-126775, Year 2020 |
| Publish date | Nov 8, 2018 (structure data deposition date) |
Authors | Furuya, N. / Momose, T. / Katsuno, K. / Fushimi, N. / Muranaka, H. / Handa, C. / Sawa, M. / Ozawa, T. / Kinoshita, T. |
External links | Bioorg. Med. Chem. Lett. / PubMed:31699609 |
| Methods | X-ray diffraction |
| Resolution | 2.54 Å |
| Structure data | ![]() PDB-6iqn: |
| Chemicals | ![]() ChemComp-AQ6: ![]() ChemComp-HOH: |
| Source |
|
Keywords | TRANSFERASE / Inhibitor |
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homo sapiens (human)
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