+Search query
-Structure paper
Title | Discovery of Small Molecule Antagonists of the USP5 Zinc Finger Ubiquitin-Binding Domain. |
---|---|
Journal, issue, pages | J. Med. Chem., Vol. 62, Page 10144-10155, Year 2019 |
Publish date | Jun 28, 2018 (structure data deposition date) |
Authors | Mann, M.K. / Franzoni, I. / de Freitas, R.F. / Tempel, W. / Houliston, S. / Smith, L. / Vedadi, M. / Arrowsmith, C.H. / Harding, R.J. / Schapira, M. |
External links | J. Med. Chem. / PubMed:31663737 |
Methods | X-ray diffraction |
Resolution | 1.65 - 2.1 Å |
Structure data | PDB-6dxh: PDB-6dxt: PDB-6nft: PDB-6p9g: |
Chemicals | ChemComp-UNX: ChemComp-ZN: ChemComp-HH4: ChemComp-HOH: ChemComp-HHY: ChemComp-EDO: ChemComp-KKG: ChemComp-O4Y: |
Source |
|
Keywords | HYDROLASE / DEUBIQUITINASE / USP5 / UBIQUITIN / STRUCTURAL GENOMICS CONSORTIUM / SGC / Structural Genomics / PROTEIN BINDING / ubiquitin binding domain |