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-Structure paper
Title | Building Bridges in a Series of Estrogen Receptor Degraders: An Application of Metathesis in Medicinal Chemistry. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 1492-1497, Year 2019 |
Publish date | Sep 3, 2019 (structure data deposition date) |
Authors | Scott, J.S. / Breed, J. / Carbajo, R.J. / Davey, P.R. / Greenwood, R. / Huynh, H.K. / Klinowska, T. / Morrow, C.J. / Moss, T.A. / Polanski, R. ...Scott, J.S. / Breed, J. / Carbajo, R.J. / Davey, P.R. / Greenwood, R. / Huynh, H.K. / Klinowska, T. / Morrow, C.J. / Moss, T.A. / Polanski, R. / Nissink, J.W.M. / Varnes, J. / Yang, B. |
External links | Acs Med. Chem. Lett. / PubMed:31620239 |
Methods | X-ray diffraction |
Resolution | 1.74 - 1.77 Å |
Structure data | PDB-6sq0: PDB-6suo: |
Chemicals | ChemComp-LRQ: ChemComp-HOH: ChemComp-LVH: |
Source |
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Keywords | GENE REGULATION / oestrogen receptor / oestrogen binding domain |