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-Structure paper
Title | Discovery of MK-8719, a Potent O-GlcNAcase Inhibitor as a Potential Treatment for Tauopathies. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 10062-10097, Year 2019 |
Publish date | Jul 1, 2019 (structure data deposition date) |
Authors | Selnick, H.G. / Hess, J.F. / Tang, C. / Liu, K. / Schachter, J.B. / Ballard, J.E. / Marcus, J. / Klein, D.J. / Wang, X. / Pearson, M. ...Selnick, H.G. / Hess, J.F. / Tang, C. / Liu, K. / Schachter, J.B. / Ballard, J.E. / Marcus, J. / Klein, D.J. / Wang, X. / Pearson, M. / Savage, M.J. / Kaul, R. / Li, T.S. / Vocadlo, D.J. / Zhou, Y. / Zhu, Y. / Mu, C. / Wang, Y. / Wei, Z. / Bai, C. / Duffy, J.L. / McEachern, E.J. |
External links | J. Med. Chem. / PubMed:31487175 |
Methods | X-ray diffraction |
Resolution | 2.86 Å |
Structure data | PDB-6pm9: |
Chemicals | ChemComp-OQ1: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / O-GLCNACASE / GH84 / INHIBITOR |