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-Structure paper
Title | Rigidification Dramatically Improves Inhibitor Selectivity for RAF Kinases. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 1074-1080, Year 2019 |
Publish date | Jan 25, 2019 (structure data deposition date) |
Authors | Assadieskandar, A. / Yu, C. / Maisonneuve, P. / Kurinov, I. / Sicheri, F. / Zhang, C. |
External links | Acs Med. Chem. Lett. / PubMed:31312411 |
Methods | X-ray diffraction |
Resolution | 3.05 Å |
Structure data | PDB-6nsq: |
Chemicals | ChemComp-KZP: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / BRAF inhibitors / SIGNALING PROTEIN / TRANSFERASE-TRANSFERASE Inhibitor complex / TRANSFERASE |