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-Structure paper
Title | Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 7146-7159, Year 2019 |
Publish date | Apr 9, 2019 (structure data deposition date) |
![]() | Leaver, D.J. / Cleary, B. / Nguyen, N. / Priebbenow, D.L. / Lagiakos, H.R. / Sanchez, J. / Xue, L. / Huang, F. / Sun, Y. / Mujumdar, P. ...Leaver, D.J. / Cleary, B. / Nguyen, N. / Priebbenow, D.L. / Lagiakos, H.R. / Sanchez, J. / Xue, L. / Huang, F. / Sun, Y. / Mujumdar, P. / Mudududdla, R. / Varghese, S. / Teguh, S. / Charman, S.A. / White, K.L. / Katneni, K. / Cuellar, M. / Strasser, J.M. / Dahlin, J.L. / Walters, M.A. / Street, I.P. / Monahan, B.J. / Jarman, K.E. / Sabroux, H.J. / Falk, H. / Chung, M.C. / Hermans, S.J. / Parker, M.W. / Thomas, T. / Baell, J.B. |
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Methods | X-ray diffraction |
Resolution | 1.7 - 2.03 Å |
Structure data | ![]() PDB-6oin: ![]() PDB-6oio: ![]() PDB-6oip: ![]() PDB-6oiq: ![]() PDB-6oir: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-MQJ: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-ML7: ![]() ChemComp-MLS: ![]() ChemComp-MLV: ![]() ChemComp-MNJ: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Inhibitor / Complex / MYST / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |