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-Structure paper
Title | Folding Then Binding vs Folding Through Binding in Macrocyclic Peptide Inhibitors of Human Pancreatic alpha-Amylase. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 14, Page 1751-1759, Year 2019 |
Publish date | Dec 1, 2016 (structure data deposition date) |
Authors | Goldbach, L. / Vermeulen, B.J.A. / Caner, S. / Liu, M. / Tysoe, C. / van Gijzel, L. / Yoshisada, R. / Trellet, M. / van Ingen, H. / Brayer, G.D. ...Goldbach, L. / Vermeulen, B.J.A. / Caner, S. / Liu, M. / Tysoe, C. / van Gijzel, L. / Yoshisada, R. / Trellet, M. / van Ingen, H. / Brayer, G.D. / Bonvin, A.M.J.J. / Jongkees, S.A.K. |
External links | Acs Chem. Biol. / PubMed:31241898 |
Methods | X-ray diffraction |
Resolution | 0.95 - 2.55 Å |
Structure data | PDB-5u3a: PDB-5va9: |
Chemicals | ChemComp-NAG: ChemComp-CL: ChemComp-CA: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / Amylase / Diabetes / Obesity / Glucosyl hydrolase / hydrolase/hydrolase inhibitor / peptide inhibitor complex / hydrolase-hydrolase inhibitor complex |