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-Structure paper
Title | Ripretinib (DCC-2618) Is a Switch Control Kinase Inhibitor of a Broad Spectrum of Oncogenic and Drug-Resistant KIT and PDGFRA Variants. |
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Journal, issue, pages | Cancer Cell, Vol. 35, Page 738-751.e9, Year 2019 |
Publish date | Oct 4, 2018 (structure data deposition date) |
![]() | Smith, B.D. / Kaufman, M.D. / Lu, W.P. / Gupta, A. / Leary, C.B. / Wise, S.C. / Rutkoski, T.J. / Ahn, Y.M. / Al-Ani, G. / Bulfer, S.L. ...Smith, B.D. / Kaufman, M.D. / Lu, W.P. / Gupta, A. / Leary, C.B. / Wise, S.C. / Rutkoski, T.J. / Ahn, Y.M. / Al-Ani, G. / Bulfer, S.L. / Caldwell, T.M. / Chun, L. / Ensinger, C.L. / Hood, M.M. / McKinley, A. / Patt, W.C. / Ruiz-Soto, R. / Su, Y. / Telikepalli, H. / Town, A. / Turner, B.A. / Vogeti, L. / Vogeti, S. / Yates, K. / Janku, F. / Abdul Razak, A.R. / Rosen, O. / Heinrich, M.C. / Flynn, D.L. |
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Methods | X-ray diffraction |
Resolution | 1.8 Å |
Structure data | ![]() PDB-6mob: |
Chemicals | ![]() ChemComp-NO3: ![]() ChemComp-JWY: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / Deciphera / Kit1 kinase / DP2976 / decode / TRANSFERASE-TRANSFERASE INHIBITOR complex |