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-Structure paper
Title | Structural and pharmacological evaluation of a novel non-nucleoside reverse transcriptase inhibitor as a promising long acting nanoformulation for treating HIV. |
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Journal, issue, pages | Antiviral Res., Vol. 167, Page 110-116, Year 2019 |
Publish date | Mar 27, 2019 (structure data deposition date) |
![]() | Kudalkar, S.N. / Ullah, I. / Bertoletti, N. / Mandl, H.K. / Cisneros, J.A. / Beloor, J. / Chan, A.H. / Quijano, E. / Saltzman, W.M. / Jorgensen, W.L. ...Kudalkar, S.N. / Ullah, I. / Bertoletti, N. / Mandl, H.K. / Cisneros, J.A. / Beloor, J. / Chan, A.H. / Quijano, E. / Saltzman, W.M. / Jorgensen, W.L. / Kumar, P. / Anderson, K.S. |
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Methods | X-ray diffraction |
Resolution | 2.9 Å |
Structure data | ![]() PDB-6oe3: |
Chemicals | ![]() ChemComp-M9A: ![]() ChemComp-MG: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / NNRTIs / HIV-1 / drug design |