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-Structure paper
Title | Identification of entacapone as a chemical inhibitor of FTO mediating metabolic regulation through FOXO1. |
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Journal, issue, pages | Sci Transl Med, Vol. 11, Year 2019 |
Publish date | Aug 5, 2018 (structure data deposition date) |
![]() | Peng, S. / Xiao, W. / Ju, D. / Sun, B. / Hou, N. / Liu, Q. / Wang, Y. / Zhao, H. / Gao, C. / Zhang, S. ...Peng, S. / Xiao, W. / Ju, D. / Sun, B. / Hou, N. / Liu, Q. / Wang, Y. / Zhao, H. / Gao, C. / Zhang, S. / Cao, R. / Li, P. / Huang, H. / Ma, Y. / Lai, W. / Ma, Z. / Zhang, W. / Huang, S. / Wang, H. / Zhang, Z. / Zhao, L. / Cai, T. / Zhao, Y.L. / Wang, F. / Nie, Y. / Zhi, G. / Yang, Y.G. / Zhang, E.E. / Huang, N. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | ![]() PDB-6aej: ![]() PDB-6ak4: |
Chemicals | ![]() ChemComp-7YC: ![]() ChemComp-ZN: ![]() ChemComp-PD9: |
Source |
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![]() | OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR / OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX / OXIDOREDUCTASE |