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-Structure paper
Title | Fragment-Based Discovery of an Apolipoprotein E4 (apoE4) Stabilizer. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 4120-4130, Year 2019 |
Publish date | Dec 11, 2018 (structure data deposition date) |
![]() | Petros, A.M. / Korepanova, A. / Jakob, C.G. / Qiu, W. / Panchal, S.C. / Wang, J. / Dietrich, J.D. / Brewer, J.T. / Pohlki, F. / Kling, A. ...Petros, A.M. / Korepanova, A. / Jakob, C.G. / Qiu, W. / Panchal, S.C. / Wang, J. / Dietrich, J.D. / Brewer, J.T. / Pohlki, F. / Kling, A. / Wilcox, K. / Lakics, V. / Bahnassawy, L. / Reinhardt, P. / Partha, S.K. / Bodelle, P.M. / Lake, M. / Charych, E.I. / Stoll, V.S. / Sun, C. / Mohler, E.G. |
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Methods | X-ray diffraction |
Resolution | 1.707 - 1.82 Å |
Structure data | ![]() PDB-6ncn: ![]() PDB-6nco: |
Chemicals | ![]() ChemComp-KJM: ![]() ChemComp-HOH: ![]() ChemComp-KQP: |
Source |
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![]() | LIPID TRANSPORT / Lipid Binding Lipid Transport / Lipid Binding |