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-Structure paper
Title | Lead optimization and efficacy evaluation of quinazoline-based BET family inhibitors for potential treatment of cancer and inflammatory diseases. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 29, Page 1220-1226, Year 2019 |
Publish date | Aug 28, 2018 (structure data deposition date) |
![]() | Yang, S.M. / Yoshioka, M. / Strovel, J.W. / Urban, D.J. / Hu, X. / Hall, M.D. / Jadhav, A. / Maloney, D.J. |
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Methods | X-ray diffraction |
Resolution | 2.11 Å |
Structure data | ![]() PDB-6mau: |
Chemicals | ![]() ChemComp-JBS: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | PROTEIN BINDING / BRD4(1) |