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-Structure paper
Title | Structure-guided design fine-tunes pharmacokinetics, tolerability, and antitumor profile of multispecific frizzled antibodies. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. U.S.A., Vol. 116, Page 6812-6817, Year 2019 |
Publish date | Feb 26, 2019 (structure data deposition date) |
![]() | Raman, S. / Beilschmidt, M. / To, M. / Lin, K. / Lui, F. / Jmeian, Y. / Ng, M. / Fernandez, M. / Fu, Y. / Mascall, K. ...Raman, S. / Beilschmidt, M. / To, M. / Lin, K. / Lui, F. / Jmeian, Y. / Ng, M. / Fernandez, M. / Fu, Y. / Mascall, K. / Duque, A. / Wang, X. / Pan, G. / Angers, S. / Moffat, J. / Sidhu, S.S. / Magram, J. / Sinclair, A.M. / Fransson, J. / Julien, J.P. |
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Methods | X-ray diffraction |
Resolution | 1.8 - 2.5 Å |
Structure data | ![]() PDB-6o39: ![]() PDB-6o3a: ![]() PDB-6o3b: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-ACT: ![]() ChemComp-NAG: ![]() ChemComp-HOH: ![]() ChemComp-CXS: ![]() ChemComp-NA: ![]() ChemComp-GOL: |
Source |
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![]() | SIGNALING PROTEIN / Receptor / Wnt / Frizzled / CRD / Antibody |