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-Structure paper
Title | Shooting three inflammatory targets with a single bullet: Novel multi-targeting anti-inflammatory glitazones. |
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Journal, issue, pages | Eur J Med Chem, Vol. 167, Page 562-582, Year 2019 |
Publish date | Jul 19, 2018 (structure data deposition date) |
![]() | Elzahhar, P.A. / Alaaeddine, R. / Ibrahim, T.M. / Nassra, R. / Ismail, A. / Chua, B.S.K. / Frkic, R.L. / Bruning, J.B. / Wallner, N. / Knape, T. ...Elzahhar, P.A. / Alaaeddine, R. / Ibrahim, T.M. / Nassra, R. / Ismail, A. / Chua, B.S.K. / Frkic, R.L. / Bruning, J.B. / Wallner, N. / Knape, T. / von Knethen, A. / Labib, H. / El-Yazbi, A.F. / Belal, A.S.F. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-6e5a: |
Chemicals | ![]() ChemComp-HV4: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / PPAR / nuclear receptor / transcription factor / ligand binding domain |