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-Structure paper
Title | Bidirectional modulation of HIF-2 activity through chemical ligands. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 15, Page 367-376, Year 2019 |
Publish date | Jul 15, 2018 (structure data deposition date) |
![]() | Wu, D. / Su, X. / Lu, J. / Li, S. / Hood, B.L. / Vasile, S. / Potluri, N. / Diao, X. / Kim, Y. / Khorasanizadeh, S. / Rastinejad, F. |
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Methods | X-ray diffraction |
Resolution | 2.85 - 3 Å |
Structure data | ![]() PDB-6e3s: ![]() PDB-6e3t: ![]() PDB-6e3u: |
Chemicals | ![]() ChemComp-79A: ![]() ChemComp-HO7: ![]() ChemComp-HNJ: |
Source |
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![]() | transcription/transcription inhibitor / Complex / Antagonist / Transcription factor / transcription-transcription inhibitor complex / transcription/agonist / Agonist / TRANSCRIPTION / transcription-agonist complex |