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-Structure paper
Title | Designing Dual Inhibitors of Anaplastic Lymphoma Kinase (ALK) and Bromodomain-4 (BRD4) by Tuning Kinase Selectivity. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 2618-2637, Year 2019 |
Publish date | Dec 4, 2018 (structure data deposition date) |
![]() | Watts, E. / Heidenreich, D. / Tucker, E. / Raab, M. / Strebhardt, K. / Chesler, L. / Knapp, S. / Bellenie, B. / Hoelder, S. |
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Methods | X-ray diffraction |
Resolution | 1.2 - 2 Å |
Structure data | ![]() PDB-6q3y: ![]() PDB-6q3z: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-HG5: ![]() ChemComp-HOH: ![]() ChemComp-HG8: |
Source |
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![]() | GENE REGULATION / BRD4(BD1) / inhibitor / complex / Structural Genomics / Structural Genomics Consortium / SGC |