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-Structure paper
| Title | A class of highly selective inhibitors bind to an active state of PI3K gamma. |
|---|---|
| Journal, issue, pages | Nat. Chem. Biol., Vol. 15, Page 348-357, Year 2019 |
| Publish date | Jun 27, 2018 (structure data deposition date) |
Authors | Gangadhara, G. / Dahl, G. / Bohnacker, T. / Rae, R. / Gunnarsson, J. / Blaho, S. / Oster, L. / Lindmark, H. / Karabelas, K. / Pemberton, N. ...Gangadhara, G. / Dahl, G. / Bohnacker, T. / Rae, R. / Gunnarsson, J. / Blaho, S. / Oster, L. / Lindmark, H. / Karabelas, K. / Pemberton, N. / Tyrchan, C. / Mogemark, M. / Wymann, M.P. / Williams, R.L. / Perry, M.W.D. / Papavoine, T. / Petersen, J. |
External links | Nat. Chem. Biol. / PubMed:30718815 |
| Methods | X-ray diffraction |
| Resolution | 2.55 Å |
| Structure data | ![]() PDB-6gy0: |
| Chemicals | ![]() ChemComp-FGE: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE / Inhibitor / PI3K |
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