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-Structure paper
Title | Suppression of Tumor Growth and Metastases by Targeted Intervention in Urokinase Activity with Cyclic Peptides. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 2172-2183, Year 2019 |
Publish date | Jul 8, 2018 (structure data deposition date) |
Authors | Wang, D. / Yang, Y. / Jiang, L. / Wang, Y. / Li, J. / Andreasen, P.A. / Chen, Z. / Huang, M. / Xu, P. |
External links | J. Med. Chem. / PubMed:30707839 |
Methods | X-ray diffraction |
Resolution | 2.489 - 2.53 Å |
Structure data | PDB-6a8g: PDB-6a8n: |
Chemicals | ChemComp-PO4: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE INHIBITOR/HYDROLASE / Peptides inhibitor / muPA / serine protease / HYDROLASE / HYDROLASE INHIBITOR-HYDROLASE complex / HYDROLASE/HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |