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Title | Design, Synthesis, and Biological Evaluation of Retinoic Acid-Related Orphan Receptor gamma t (ROR gamma t) Agonist Structure-Based Functionality Switching Approach from In House ROR gamma t Inverse Agonist to ROR gamma t Agonist. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 1167-1179, Year 2019 |
Publish date | Jul 13, 2018 (structure data deposition date) |
Authors | Yukawa, T. / Nara, Y. / Kono, M. / Sato, A. / Oda, T. / Takagi, T. / Sato, T. / Banno, Y. / Taya, N. / Imada, T. ...Yukawa, T. / Nara, Y. / Kono, M. / Sato, A. / Oda, T. / Takagi, T. / Sato, T. / Banno, Y. / Taya, N. / Imada, T. / Shiokawa, Z. / Negoro, N. / Kawamoto, T. / Koyama, R. / Uchiyama, N. / Skene, R. / Hoffman, I. / Chen, C.H. / Sang, B. / Snell, G. / Katsuyama, R. / Yamamoto, S. / Shirai, J. |
External links | J. Med. Chem. / PubMed:30652849 |
Methods | X-ray diffraction |
Resolution | 2.1 - 2.47 Å |
Structure data | PDB-6e3e: PDB-6e3g: |
Chemicals | ChemComp-SO4: ChemComp-MPD: ChemComp-HQ7: ChemComp-HOH: ChemComp-EDO: ChemComp-HOJ: |
Source |
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Keywords | nuclear protein/agonist / Nuclear hormone receptor / inverse agonist / nuclear protein-agonist complex / agonist / NUCLEAR PROTEIN |