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Title | Iterative Design and Optimization of Initially Inactive Proteolysis Targeting Chimeras (PROTACs) Identify VZ185 as a Potent, Fast, and Selective von Hippel-Lindau (VHL) Based Dual Degrader Probe of BRD9 and BRD7. |
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Journal, issue, pages | J. Med. Chem., Vol. 62, Page 699-726, Year 2019 |
Publish date | Sep 11, 2018 (structure data deposition date) |
![]() | Zoppi, V. / Hughes, S.J. / Maniaci, C. / Testa, A. / Gmaschitz, T. / Wieshofer, C. / Koegl, M. / Riching, K.M. / Daniels, D.L. / Spallarossa, A. / Ciulli, A. |
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Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-6hm0: |
Chemicals | ![]() ChemComp-GBW: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / PROTAC / LYSINE-ACETYLATED HISTONE BINDING / CHROMATIN REGULATOR |