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-Structure paper
| Title | Molecular mechanism of a covalent allosteric inhibitor of SUMO E1 activating enzyme. |
|---|---|
| Journal, issue, pages | Nat Commun, Vol. 9, Page 5145-5145, Year 2018 |
| Publish date | Apr 1, 2018 (structure data deposition date) |
Authors | Lv, Z. / Yuan, L. / Atkison, J.H. / Williams, K.M. / Vega, R. / Sessions, E.H. / Divlianska, D.B. / Davies, C. / Chen, Y. / Olsen, S.K. |
External links | Nat Commun / PubMed:30514846 |
| Methods | X-ray diffraction |
| Resolution | 2.462 - 3.1 Å |
| Structure data | ![]() PDB-6cwy: ![]() PDB-6cwz: |
| Chemicals | ![]() ChemComp-GOL: ![]() ChemComp-ZN: ![]() ChemComp-MG: ![]() ChemComp-SO4: ![]() ChemComp-FHJ: ![]() ChemComp-HOH: |
| Source |
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Keywords | transferase/transferase inhibitor / ROSSMANN-LIKE FOLD / UBIQUITIN-LIKE FOLD / UBIQUITIN ACTIVATING ENZYME / ACTIVITY / ATP BINDING / LIGASE ACTIVITY / ATP/MG BINDING / UBIQUITIN E2 / LIGASE / TRANSFERASE / transferase-transferase inhibitor complex |
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