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-Structure paper
Title | The SERM/SERD bazedoxifene disrupts ESR1 helix 12 to overcome acquired hormone resistance in breast cancer cells. |
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Journal, issue, pages | Elife, Vol. 7, Year 2018 |
Publish date | Jan 6, 2015 (structure data deposition date) |
![]() | Fanning, S.W. / Jeselsohn, R. / Dharmarajan, V. / Mayne, C.G. / Karimi, M. / Buchwalter, G. / Houtman, R. / Toy, W. / Fowler, C.E. / Han, R. ...Fanning, S.W. / Jeselsohn, R. / Dharmarajan, V. / Mayne, C.G. / Karimi, M. / Buchwalter, G. / Houtman, R. / Toy, W. / Fowler, C.E. / Han, R. / Laine, M. / Carlson, K.E. / Martin, T.A. / Nowak, J. / Nwachukwu, J.C. / Hosfield, D.J. / Chandarlapaty, S. / Tajkhorshid, E. / Nettles, K.W. / Griffin, P.R. / Shen, Y. / Katzenellenbogen, J.A. / Brown, M. / Greene, G.L. |
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Methods | X-ray diffraction |
Resolution | 2.491 Å |
Structure data | ![]() PDB-4xi3: |
Chemicals | ![]() ChemComp-29S: ![]() ChemComp-HOH: |
Source |
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![]() | SIGNALING PROTEIN / Estrogen Receptor / SERM / Bazedoxifene / Breast Cancer / Nuclear Hormone Receptor |