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-Structure paper
| Title | Discovery of a novel azetidine scaffold for colony stimulating factor-1 receptor (CSF-1R) Type II inhibitors by the use of docking models. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 29, Page 115-118, Year 2019 |
| Publish date | Sep 25, 2018 (structure data deposition date) |
Authors | Ikegashira, K. / Ikenogami, T. / Yamasaki, T. / Hase, Y. / Yamaguchi, T. / Inagaki, K. / Doi, S. / Adachi, T. / Koga, Y. / Hashimoto, H. |
External links | Bioorg. Med. Chem. Lett. / PubMed:30442420 |
| Methods | X-ray diffraction |
| Resolution | 1.8 Å |
| Structure data | ![]() PDB-6ig8: |
| Chemicals | ![]() ChemComp-MG: ![]() ChemComp-GOL: ![]() ChemComp-A7O: ![]() ChemComp-HOH: |
| Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / CSF-1-R / FMS PROTO-ONCOGENE / C-FMS / CD115 antigen / Kinase / ATP-binding / TRANSFERASE-TRANSFERASE INHIBITOR complex |
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homo sapiens (human)
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