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Title | Aurora A Kinase Inhibition Is Synthetic Lethal with Loss of theRB1Tumor Suppressor Gene. |
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Journal, issue, pages | Cancer Discov, Vol. 9, Page 248-263, Year 2019 |
Publish date | Jan 8, 2018 (structure data deposition date) |
Authors | Gong, X. / Du, J. / Parsons, S.H. / Merzoug, F.F. / Webster, Y. / Iversen, P.W. / Chio, L.C. / Van Horn, R.D. / Lin, X. / Blosser, W. ...Gong, X. / Du, J. / Parsons, S.H. / Merzoug, F.F. / Webster, Y. / Iversen, P.W. / Chio, L.C. / Van Horn, R.D. / Lin, X. / Blosser, W. / Han, B. / Jin, S. / Yao, S. / Bian, H. / Ficklin, C. / Fan, L. / Kapoor, A. / Antonysamy, S. / Mc Nulty, A.M. / Froning, K. / Manglicmot, D. / Pustilnik, A. / Weichert, K. / Wasserman, S.R. / Dowless, M. / Marugan, C. / Baquero, C. / Lallena, M.J. / Eastman, S.W. / Hui, Y.H. / Dieter, M.Z. / Doman, T. / Chu, S. / Qian, H.R. / Ye, X.S. / Barda, D.A. / Plowman, G.D. / Reinhard, C. / Campbell, R.M. / Henry, J.R. / Buchanan, S.G. |
External links | Cancer Discov / PubMed:30373917 |
Methods | X-ray diffraction |
Resolution | 1.73 - 1.96 Å |
Structure data | PDB-6c2r: PDB-6c2t: |
Chemicals | ChemComp-SO4: ChemComp-EG7: ChemComp-HOH: ChemComp-EGJ: ChemComp-DMS: |
Source |
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Keywords | TRANSFERASE / Protein kinase |