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-Structure paper
Title | Small molecule inhibitors reveal allosteric regulation of USP14 via steric blockade. |
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Journal, issue, pages | Cell Res., Vol. 28, Page 1186-1194, Year 2018 |
Publish date | Oct 6, 2018 (structure data deposition date) |
![]() | Wang, Y. / Jiang, Y. / Ding, S. / Li, J. / Song, N. / Ren, Y. / Hong, D. / Wu, C. / Li, B. / Wang, F. ...Wang, Y. / Jiang, Y. / Ding, S. / Li, J. / Song, N. / Ren, Y. / Hong, D. / Wu, C. / Li, B. / Wang, F. / He, W. / Wang, J. / Mei, Z. |
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Methods | X-ray diffraction |
Resolution | 1.97 - 2.53 Å |
Structure data | ![]() PDB-6iik: ![]() PDB-6iil: ![]() PDB-6iim: ![]() PDB-6iin: |
Chemicals | ![]() ChemComp-IU1: ![]() ChemComp-HOH: ![]() ChemComp-A8F: ![]() ChemComp-A8L: ![]() ChemComp-A8O: |
Source |
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![]() | HYDROLASE / USP14 inhibitor complex / STRUCTURAL PROTEIN |