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Title | Design, synthesis, and evaluation of cystargolide-based beta-lactones as potent proteasome inhibitors. |
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Journal, issue, pages | Eur J Med Chem, Vol. 157, Page 962-977, Year 2018 |
Publish date | Apr 5, 2018 (structure data deposition date) |
![]() | Niroula, D. / Hallada, L.P. / Le Chapelain, C. / Ganegamage, S.K. / Dotson, D. / Rogelj, S. / Groll, M. / Tello-Aburto, R. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.7 - 3 Å |
Structure data | ![]() PDB-6g7f: ![]() PDB-6g8m: ![]() PDB-6g8n: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-CL: ![]() ChemComp-EPW: ![]() ChemComp-HOH: ![]() ChemComp-EQE: ![]() ChemComp-EQB: |
Source |
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![]() | HYDROLASE / Proteasome / Inhibitor / Beta Lactone; Natural Product / Binding Analysis / Beta Lactone; Natural Product Derivative |