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-Structure paper
Title | Amelioration of PXR-mediated CYP3A4 induction by mGluR2 modulators. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 28, Page 3194-3196, Year 2018 |
Publish date | Jun 21, 2018 (structure data deposition date) |
![]() | Vaz, R.J. / Li, Y. / Chellaraj, V. / Reiling, S. / Kuntzweiler, T. / Yang, D. / Shen, H. / Batchelor, J.D. / Zhang, Y. / Chen, X. ...Vaz, R.J. / Li, Y. / Chellaraj, V. / Reiling, S. / Kuntzweiler, T. / Yang, D. / Shen, H. / Batchelor, J.D. / Zhang, Y. / Chen, X. / McLean, L.R. / Kosley Jr., R. |
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Methods | X-ray diffraction |
Resolution | 2.3 Å |
Structure data | ![]() PDB-6dup: |
Chemicals | ![]() ChemComp-HCJ: ![]() ChemComp-HOH: |
Source |
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![]() | NUCLEAR PROTEIN / PXR |