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-Structure paper
Title | A Novel, Nonpeptidic, Orally Active Bivalent Inhibitor of Human beta-Tryptase. |
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Journal, issue, pages | Pharmacology, Vol. 102, Page 233-243, Year 2018 |
Publish date | Sep 13, 2013 (structure data deposition date) |
![]() | Giardina, S.F. / Werner, D.S. / Pingle, M. / Bergstrom, D.E. / Arnold, L.D. / Barany, F. |
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Methods | X-ray diffraction |
Resolution | 1.95 Å |
Structure data | ![]() PDB-4mpw: |
Chemicals | ![]() ChemComp-CL: ![]() ChemComp-PGE: ![]() ChemComp-ACT: ![]() ChemComp-2AJ: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / coferon / alpha-hydroxyketone / small molecule inhibitor / drug discovery / self-assembly / crystal catalysis / silanol / HYDROLASE-HYDROLASE INHIBITOR complex |