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-Structure paper
Title | ROCK inhibitors 2. Improving potency, selectivity and solubility through the application of rationally designed solubilizing groups. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Year 2018 |
Publish date | Jan 28, 2016 (structure data deposition date) |
Authors | Gao, H. / Marhefka, C. / Jacobs, M.D. / Cao, J. / Bandarage, U.K. / Green, J. |
External links | Bioorg. Med. Chem. Lett. / PubMed:29945794 |
Methods | X-ray diffraction |
Resolution | 2.8 Å |
Structure data | PDB-5hvu: |
Chemicals | ChemComp-65R: ChemComp-HOH: |
Source |
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Keywords | Transferase/transferase inhibitor / kinase / inhibitor / complex / solubilizing group / Transferase-transferase inhibitor complex |