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-Structure paper
Title | An Unusual Intramolecular Halogen Bond Guides Conformational Selection. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 57, Page 9970-9975, Year 2018 |
Publish date | May 29, 2018 (structure data deposition date) |
Authors | Tesch, R. / Becker, C. / Muller, M.P. / Beck, M.E. / Quambusch, L. / Getlik, M. / Lategahn, J. / Uhlenbrock, N. / Costa, F.N. / Poleto, M.D. ...Tesch, R. / Becker, C. / Muller, M.P. / Beck, M.E. / Quambusch, L. / Getlik, M. / Lategahn, J. / Uhlenbrock, N. / Costa, F.N. / Poleto, M.D. / Pinheiro, P.S.M. / Rodrigues, D.A. / Sant'Anna, C.M.R. / Ferreira, F.F. / Verli, H. / Fraga, C.A.M. / Rauh, D. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:29873877 |
Methods | X-ray diffraction |
Resolution | 2.6 Å |
Structure data | PDB-6gn1: |
Chemicals | ChemComp-CL: ChemComp-F4N: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / Glycogen synthase kinase-3 beta / PIK-75 / halogen bond / inhibitor |