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-Structure paper
Title | Unbiased Combinatorial Screening Identifies a Bispecific IgG1 that Potently Inhibits HER3 Signaling via HER2-Guided Ligand Blockade. |
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Journal, issue, pages | Cancer Cell, Vol. 33, Page 922-936.e10, Year 2018 |
Publish date | May 29, 2017 (structure data deposition date) |
![]() | Geuijen, C.A.W. / De Nardis, C. / Maussang, D. / Rovers, E. / Gallenne, T. / Hendriks, L.J.A. / Visser, T. / Nijhuis, R. / Logtenberg, T. / de Kruif, J. ...Geuijen, C.A.W. / De Nardis, C. / Maussang, D. / Rovers, E. / Gallenne, T. / Hendriks, L.J.A. / Visser, T. / Nijhuis, R. / Logtenberg, T. / de Kruif, J. / Gros, P. / Throsby, M. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 3 - 4.5 Å |
Structure data | ![]() PDB-5o4g: ![]() PDB-5o4o: ![]() PDB-5o7p: |
Chemicals | ![]() ChemComp-NAG: |
Source |
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![]() | ONCOPROTEIN / HER2 ectodomain / complex / Fab / transferase / IMMUNE SYSTEM / HER3 ectodomain |