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-Structure paper
Title | TP-064, a potent and selective small molecule inhibitor of PRMT4 for multiple myeloma. |
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Journal, issue, pages | Oncotarget, Vol. 9, Page 18480-18493, Year 2018 |
Publish date | Dec 6, 2016 (structure data deposition date) |
![]() | Nakayama, K. / Szewczyk, M.M. / Dela Sena, C. / Wu, H. / Dong, A. / Zeng, H. / Li, F. / de Freitas, R.F. / Eram, M.S. / Schapira, M. ...Nakayama, K. / Szewczyk, M.M. / Dela Sena, C. / Wu, H. / Dong, A. / Zeng, H. / Li, F. / de Freitas, R.F. / Eram, M.S. / Schapira, M. / Baba, Y. / Kunitomo, M. / Cary, D.R. / Tawada, M. / Ohashi, A. / Imaeda, Y. / Saikatendu, K.S. / Grimshaw, C.E. / Vedadi, M. / Arrowsmith, C.H. / Barsyte-Lovejoy, D. / Kiba, A. / Tomita, D. / Brown, P.J. |
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Methods | X-ray diffraction |
Resolution | 1.88 Å |
Structure data | ![]() PDB-5u4x: |
Chemicals | ![]() ChemComp-SAH: ![]() ChemComp-7VM: ![]() ChemComp-UNX: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / CARM1 / methyltransferase / TP-064 / Structural Genomics / Structural Genomics Consortium / SGC |