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-Structure paper
Title | An orally available, brain-penetrant CAMKK2 inhibitor reduces food intake in rodent model. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 28, Page 1958-1963, Year 2018 |
Publish date | Mar 5, 2018 (structure data deposition date) |
![]() | Price, D.J. / Drewry, D.H. / Schaller, L.T. / Thompson, B.D. / Reid, P.R. / Maloney, P.R. / Liang, X. / Banker, P. / Buckholz, R.G. / Selley, P.K. ...Price, D.J. / Drewry, D.H. / Schaller, L.T. / Thompson, B.D. / Reid, P.R. / Maloney, P.R. / Liang, X. / Banker, P. / Buckholz, R.G. / Selley, P.K. / McDonald, O.B. / Smith, J.L. / Shearer, T.W. / Cox, R.F. / Williams, S.P. / Reid, R.A. / Tacconi, S. / Faggioni, F. / Piubelli, C. / Sartori, I. / Tessari, M. / Wang, T.Y. |
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Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-6cmj: |
Chemicals | ![]() ChemComp-F6J: ![]() ChemComp-FMT: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/TRANSFERASE INHIBITOR / kinase / signaling protein / TRANSFERASE-TRANSFERASE INHIBITOR complex |