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-Structure paper
| Title | Identification and biological evaluation of thiazole-based inverse agonists of ROR gamma t. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 28, Page 1446-1455, Year 2018 |
| Publish date | Mar 28, 2018 (structure data deposition date) |
Authors | Gege, C. / Cummings, M.D. / Albers, M. / Kinzel, O. / Kleymann, G. / Schluter, T. / Steeneck, C. / Nelen, M.I. / Milligan, C. / Spurlino, J. ...Gege, C. / Cummings, M.D. / Albers, M. / Kinzel, O. / Kleymann, G. / Schluter, T. / Steeneck, C. / Nelen, M.I. / Milligan, C. / Spurlino, J. / Xue, X. / Leonard, K. / Edwards, J.P. / Fourie, A. / Goldberg, S.D. / Hoffmann, T. |
External links | Bioorg. Med. Chem. Lett. / PubMed:29631962 |
| Methods | X-ray diffraction |
| Resolution | 3.5 Å |
| Structure data | ![]() PDB-6cvh: |
| Chemicals | ![]() ChemComp-FJG: |
| Source |
|
Keywords | NUCLEAR PROTEIN / Nuclear Receptor RORgt |
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