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-Structure paper
Title | Identification and biological evaluation of thiazole-based inverse agonists of ROR gamma t. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 28, Page 1446-1455, Year 2018 |
Publish date | Mar 28, 2018 (structure data deposition date) |
Authors | Gege, C. / Cummings, M.D. / Albers, M. / Kinzel, O. / Kleymann, G. / Schluter, T. / Steeneck, C. / Nelen, M.I. / Milligan, C. / Spurlino, J. ...Gege, C. / Cummings, M.D. / Albers, M. / Kinzel, O. / Kleymann, G. / Schluter, T. / Steeneck, C. / Nelen, M.I. / Milligan, C. / Spurlino, J. / Xue, X. / Leonard, K. / Edwards, J.P. / Fourie, A. / Goldberg, S.D. / Hoffmann, T. |
External links | Bioorg. Med. Chem. Lett. / PubMed:29631962 |
Methods | X-ray diffraction |
Resolution | 3.5 Å |
Structure data | PDB-6cvh: |
Chemicals | ChemComp-FJG: |
Source |
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Keywords | NUCLEAR PROTEIN / Nuclear Receptor RORgt |