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-Structure paper
Title | Potent 1,2,4-Triazino[5,6 b]indole-3-thioether Inhibitors of the Kanamycin Resistance Enzyme Eis from Mycobacterium tuberculosis. |
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Journal, issue, pages | ACS Infect Dis, Vol. 4, Page 1030-1040, Year 2018 |
Publish date | Sep 24, 2017 (structure data deposition date) |
![]() | Ngo, H.X. / Green, K.D. / Gajadeera, C.S. / Willby, M.J. / Holbrook, S.Y.L. / Hou, C. / Garzan, A. / Mayhoub, A.S. / Posey, J.E. / Tsodikov, O.V. / Garneau-Tsodikova, S. |
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Methods | X-ray diffraction |
Resolution | 2.4 Å |
Structure data | ![]() PDB-6b3t: |
Chemicals | ![]() ChemComp-COA: ![]() ChemComp-CJ7: ![]() ChemComp-NA: ![]() ChemComp-SO4: ![]() ChemComp-HOH: |
Source |
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![]() | transferase/transferase inhibitor / TRANSFERASE / tuberculosis / aminoglycoside / resistance / transferase-transferase inhibitor complex |