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-Structure paper
Title | Structure-based optimization of a series of selective BET inhibitors containing aniline or indoline groups. |
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Journal, issue, pages | Eur. J. Med. Chem., Vol. 150, Page 156-175, Year 2018 |
Publish date | Oct 31, 2017 (structure data deposition date) |
Authors | Hu, J. / Wang, Y. / Li, Y. / Cao, D. / Xu, L. / Song, S. / Damaneh, M.S. / Li, J. / Chen, Y. / Wang, X. ...Hu, J. / Wang, Y. / Li, Y. / Cao, D. / Xu, L. / Song, S. / Damaneh, M.S. / Li, J. / Chen, Y. / Wang, X. / Chen, L. / Shen, J. / Miao, Z. / Xiong, B. |
External links | Eur. J. Med. Chem. / PubMed:29525435 |
Methods | X-ray diffraction |
Resolution | 1.451 Å |
Structure data | PDB-5yov: |
Chemicals | ChemComp-8XR: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION/INHIBITOR / bromodomain / TRANSCRIPTION-INHIBITOR complex |