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Title | Trifunctional High-Throughput Screen Identifies Promising Scaffold To Inhibit Grp94 and Treat Myocilin-Associated Glaucoma. |
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Journal, issue, pages | ACS Chem. Biol., Vol. 13, Page 933-941, Year 2018 |
Publish date | Aug 25, 2017 (structure data deposition date) |
![]() | Huard, D.J.E. / Crowley, V.M. / Du, Y. / Cordova, R.A. / Sun, Z. / Tomlin, M.O. / Dickey, C.A. / Koren, J. / Blair, L. / Fu, H. ...Huard, D.J.E. / Crowley, V.M. / Du, Y. / Cordova, R.A. / Sun, Z. / Tomlin, M.O. / Dickey, C.A. / Koren, J. / Blair, L. / Fu, H. / Blagg, B.S.J. / Lieberman, R.L. |
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Methods | X-ray diffraction |
Resolution | 2.35 - 2.696 Å |
Structure data | ![]() PDB-6asp: ![]() PDB-6asq: |
Chemicals | ![]() ChemComp-P33: ![]() ChemComp-GOL: ![]() ChemComp-V2C: ![]() ChemComp-HOH: ![]() ChemComp-PE8: ![]() ChemComp-PEG: ![]() ChemComp-VC4: |
Source |
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![]() | CHAPERONE/INHIBITOR / Grp94 / Hsp90 / Inhibitor / Glaucoma / CHAPERONE-INHIBITOR complex |