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-Structure paper
Title | Phenylboronic Acid Derivatives as Validated Leads Active in Clinical Strains Overexpressing KPC-2: A Step against Bacterial Resistance. |
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Journal, issue, pages | Chemmedchem, Vol. 13, Page 713-724, Year 2018 |
Publish date | Jul 26, 2016 (structure data deposition date) |
![]() | Celenza, G. / Vicario, M. / Bellio, P. / Linciano, P. / Perilli, M. / Oliver, A. / Blazquez, J. / Cendron, L. / Tondi, D. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.4 - 1.5 Å |
Structure data | ![]() PDB-5ll7: ![]() PDB-5mgi: |
Chemicals | ![]() ChemComp-6YV: ![]() ChemComp-EDO: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / carbapenemase / beta-lactamase / phenyl boronic inhibitor |