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-Structure paper
Title | Discovery of Bisubstrate Inhibitors of Nicotinamide N-Methyltransferase (NNMT). |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 1541-1551, Year 2018 |
Publish date | Feb 22, 2018 (structure data deposition date) |
Authors | Babault, N. / Allali-Hassani, A. / Li, F. / Fan, J. / Yue, A. / Ju, K. / Liu, F. / Vedadi, M. / Liu, J. / Jin, J. |
External links | J. Med. Chem. / PubMed:29320176 |
Methods | X-ray diffraction |
Resolution | 2.3 Å |
Structure data | PDB-6chh: |
Chemicals | ChemComp-F0P: ChemComp-EDO: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / protein-small molecule bisubstrate inhibitor complex / TRANSFERASE / TRANSFERASE-TRANSFERASE INHIBITOR complex |