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-Structure paper
| Title | Design, synthesis, and evaluation of novel inhibitors for wild-type human serine racemase. |
|---|---|
| Journal, issue, pages | Bioorg. Med. Chem. Lett., Year 2017 |
| Publish date | Feb 1, 2017 (structure data deposition date) |
Authors | Takahara, S. / Nakagawa, K. / Uchiyama, T. / Yoshida, T. / Matsumoto, K. / Kawasumi, Y. / Mizuguchi, M. / Obita, T. / Watanabe, Y. / Hayakawa, D. ...Takahara, S. / Nakagawa, K. / Uchiyama, T. / Yoshida, T. / Matsumoto, K. / Kawasumi, Y. / Mizuguchi, M. / Obita, T. / Watanabe, Y. / Hayakawa, D. / Gouda, H. / Mori, H. / Toyooka, N. |
External links | Bioorg. Med. Chem. Lett. / PubMed:29277459 |
| Methods | X-ray diffraction |
| Resolution | 1.806 Å |
| Structure data | ![]() PDB-5x2l: |
| Chemicals | ![]() ChemComp-PLP: ![]() ChemComp-MG: ![]() ChemComp-HOH: |
| Source |
|
Keywords | LYASE / ISOMERASE / Serine Racemase / PYRIDOXAL-5'-PHOSPHATE / human |
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homo sapiens (human)
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