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-Structure paper
Title | Structure-guided design, synthesis and evaluation of oxazolidinone-based inhibitors of norovirus 3CL protease. |
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Journal, issue, pages | Eur J Med Chem, Vol. 143, Page 881-890, Year 2017 |
Publish date | Jul 10, 2017 (structure data deposition date) |
![]() | Damalanka, V.C. / Kim, Y. / Galasiti Kankanamalage, A.C. / Rathnayake, A.D. / Mehzabeen, N. / Battaile, K.P. / Lovell, S. / Nguyen, H.N. / Lushington, G.H. / Chang, K.O. / Groutas, W.C. |
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Methods | X-ray diffraction |
Resolution | 1.95 Å |
Structure data | ![]() PDB-5wej: |
Chemicals | ![]() ChemComp-V45: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE inhibitor / PROTEASE / NOROVIRUS / NORWALK VIRUS / ANTIVIRAL INHIBITORS / Oxazolidinone-based DIPEPTIDYL INHIBITOR / HYDROLASE-HYDROLASE inhibitor complex |