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Title | Discovery of Peptidomimetic Antibody-Drug Conjugate Linkers with Enhanced Protease Specificity. |
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Journal, issue, pages | J. Med. Chem., Vol. 61, Page 989-1000, Year 2018 |
Publish date | Sep 7, 2017 (structure data deposition date) |
Authors | Wei, B. / Gunzner-Toste, J. / Yao, H. / Wang, T. / Wang, J. / Xu, Z. / Chen, J. / Wai, J. / Nonomiya, J. / Tsai, S.P. ...Wei, B. / Gunzner-Toste, J. / Yao, H. / Wang, T. / Wang, J. / Xu, Z. / Chen, J. / Wai, J. / Nonomiya, J. / Tsai, S.P. / Chuh, J. / Kozak, K.R. / Liu, Y. / Yu, S.F. / Lau, J. / Li, G. / Phillips, G.D. / Leipold, D. / Kamath, A. / Su, D. / Xu, K. / Eigenbrot, C. / Steinbacher, S. / Ohri, R. / Raab, H. / Staben, L.R. / Zhao, G. / Flygare, J.A. / Pillow, T.H. / Verma, V. / Masterson, L.A. / Howard, P.W. / Safina, B. |
External links | J. Med. Chem. / PubMed:29227683 |
Methods | X-ray diffraction |
Resolution | 1.6 Å |
Structure data | PDB-6ay2: |
Chemicals | ChemComp-C1G: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE/HYDROLASE INHIBITOR / protease / covalent / inhibitor / HYDROLASE-HYDROLASE INHIBITOR complex |