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-Structure paper
Title | Discovery, optimization and biological evaluation for novel c-Met kinase inhibitors |
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Journal, issue, pages | Eur J Med Chem, Vol. 143, Page 491-502, Year 2018 |
Publish date | Aug 30, 2017 (structure data deposition date) |
Authors | Yuan, H. / Liu, Q. / Zhang, L. / Hu, S. / Chen, T. / Li, H. / Chen, Y. / Xu, Y. / Lu, T. |
External links | Eur J Med Chem / PubMed:29202410 |
Methods | X-ray diffraction |
Resolution | 1.89 Å |
Structure data | PDB-5ya5: |
Chemicals | ChemComp-6TD: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/INHIBITOR / c-MET inhibitor / TRANSFERASE-INHIBITOR complex |