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-Structure paper
Title | Design and synthesis of a biaryl series as inhibitors for the bromodomains of CBP/P300. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 28, Page 15-23, Year 2018 |
Publish date | Aug 7, 2017 (structure data deposition date) |
![]() | Lai, K.W. / Romero, F.A. / Tsui, V. / Beresini, M.H. / de Leon Boenig, G. / Bronner, S.M. / Chen, K. / Chen, Z. / Choo, E.F. / Crawford, T.D. ...Lai, K.W. / Romero, F.A. / Tsui, V. / Beresini, M.H. / de Leon Boenig, G. / Bronner, S.M. / Chen, K. / Chen, Z. / Choo, E.F. / Crawford, T.D. / Cyr, P. / Kaufman, S. / Li, Y. / Liao, J. / Liu, W. / Ly, J. / Murray, J. / Shen, W. / Wai, J. / Wang, F. / Zhu, C. / Zhu, X. / Magnuson, S. |
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Methods | X-ray diffraction |
Resolution | 1.391 Å |
Structure data | ![]() PDB-6alc: |
Chemicals | ![]() ChemComp-DMS: ![]() ChemComp-EDO: ![]() ChemComp-BKD: ![]() ChemComp-HOH: |
Source |
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![]() | PROTEIN BINDING/INHIBITOR / ![]() ![]() |