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-Structure paper
Title | Small-molecule inhibition of TLR8 through stabilization of its resting state |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 14, Page 58-64, Year 2018 |
Publish date | Jan 16, 2017 (structure data deposition date) |
Authors | Zhang, S. / Hu, Z. / Tanji, H. / Jiang, S. / Das, N. / Li, J. / Sakaniwa, K. / Jin, J. / Bian, Y. / Ohto, U. ...Zhang, S. / Hu, Z. / Tanji, H. / Jiang, S. / Das, N. / Li, J. / Sakaniwa, K. / Jin, J. / Bian, Y. / Ohto, U. / Shimizu, T. / Yin, H. |
External links | Nat. Chem. Biol. / PubMed:29155428 |
Methods | X-ray diffraction |
Resolution | 2.3 - 2.4 Å |
Structure data | PDB-5wyx: PDB-5wyz: |
Chemicals | ChemComp-NAG: ChemComp-CU8: ChemComp-HOH: ChemComp-7VF: |
Source |
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Keywords | IMMUNE SYSTEM |