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-Structure paper
Title | The X-Ray Crystal Structure of the Human Mono-Oxygenase Cytochrome P450 3A5-Ritonavir Complex Reveals Active Site Differences between P450s 3A4 and 3A5. |
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Journal, issue, pages | Mol. Pharmacol., Vol. 93, Page 14-24, Year 2018 |
Publish date | Apr 5, 2017 (structure data deposition date) |
![]() | Hsu, M.H. / Savas, U. / Johnson, E.F. |
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Methods | X-ray diffraction |
Resolution | 2.91 Å |
Structure data | ![]() PDB-5veu: |
Chemicals | ![]() ChemComp-HEM: ![]() ChemComp-RIT: |
Source |
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![]() | OXIDOREDUCTASE/OXIDOREDUCTASE inhibitor / Inhibitor / Complex / Cytochrome P450 / ritonavir / CYP3A5 / OXIDOREDUCTASE-OXIDOREDUCTASE inhibitor complex |