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-Structure paper
Title | Discovery of novel BET inhibitors by drug repurposing of nitroxoline and its analogues. |
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Journal, issue, pages | Org. Biomol. Chem., Vol. 15, Page 9352-9361, Year 2017 |
Publish date | Jul 21, 2017 (structure data deposition date) |
Authors | Jiang, H. / Xing, J. / Wang, C. / Zhang, H. / Yue, L. / Wan, X. / Chen, W. / Ding, H. / Xie, Y. / Tao, H. ...Jiang, H. / Xing, J. / Wang, C. / Zhang, H. / Yue, L. / Wan, X. / Chen, W. / Ding, H. / Xie, Y. / Tao, H. / Chen, Z. / Chen, K. / Chen, S. / Zheng, M. / Zhang, Y. / Luo, C. |
External links | Org. Biomol. Chem. / PubMed:29087414 |
Methods | X-ray diffraction |
Resolution | 1.912 Å |
Structure data | PDB-5y1y: |
Chemicals | ChemComp-HNQ: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / BRD4 inhibitor Approved drugs |