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-Structure paper
Title | D4 dopamine receptor high-resolution structures enable the discovery of selective agonists. |
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Journal, issue, pages | Science, Vol. 358, Page 381-386, Year 2017 |
Publish date | Jul 20, 2017 (structure data deposition date) |
![]() | Wang, S. / Wacker, D. / Levit, A. / Che, T. / Betz, R.M. / McCorvy, J.D. / Venkatakrishnan, A.J. / Huang, X.P. / Dror, R.O. / Shoichet, B.K. / Roth, B.L. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.962 - 2.143 Å |
Structure data | ![]() PDB-5wiu: ![]() PDB-5wiv: |
Chemicals | ![]() ChemComp-AQD: ![]() ChemComp-PO4: ![]() ChemComp-OLA: ![]() ChemComp-PEG: ![]() ChemComp-GOL: ![]() ChemComp-HOH: ![]() ChemComp-NA: |
Source |
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![]() | SIGNALING PROTEIN/ANTAGONIST / GPCR / dopamine receptor / antagonist / sodium / SIGNALING PROTEIN-ANTAGONIST complex |